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Palbociclib
來源:互聯網

Palbociclib (PD-0332991) is an orally available pyrido嘧啶derived cyclin-dependent kinase (CDK) inhibitor with potential antineoplastic activity. Palbociclib is a highly specific inhibitor of cyclindependent kinase 4 (Cdk4) (IC50, 0.011 μmol/L) and Cdk6 (IC50, 0.016 μmol/L), having no activity against a panel of 36 additional protein kinases.

化學信息

外觀:黃色至灰白色晶狀固體

分子量 : 447.53

分子式: C24H29N7O2

CAS號: 571190-30-2

溶劑/溶解度 : DMSO

晶型:2種,A和B,均為無水晶體

儲存條件: 參考CoA中推薦的條件進行儲存。

臨床信息

參考資料 >

medchemexpress.medchemexpress.cn.2015-04-27

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