來源:互聯網
Palbociclib (PD-0332991) is an orally available pyrido嘧啶derived cyclin-dependent kinase (CDK) inhibitor with potential antineoplastic activity. Palbociclib is a highly specific inhibitor of cyclindependent kinase 4 (Cdk4) (IC50, 0.011 μmol/L) and Cdk6 (IC50, 0.016 μmol/L), having no activity against a panel of 36 additional protein kinases.
化學信息
外觀:黃色至灰白色晶狀固體
分子量 : 447.53
分子式: C24H29N7O2
CAS號: 571190-30-2
晶型:2種,A和B,均為無水晶體
儲存條件: 參考CoA中推薦的條件進行儲存。
臨床信息
參考資料 >
medchemexpress.medchemexpress.cn.2015-04-27